• Akı, ;  Yalçın,  İ.;  Yıldız,  İ.;  Temiz-Arpacı,  Ö.;  Bolelli,  K.; Ertan-Bolelli, T.  DNA-Topoisomerase Inhibitory Activity of Some Heterocyclic Compounds and Their Structure-Activity Relationships. Med. Chem. Res. 2010, Suppl.: 1, 19, S6

 

  • Ceylan-Ünlüsoy, M.; Verspohl, E.J.; Ertan, R. Synthesis and antidiabetic activity of some new chromonyl-2,4-thiazolidinediones. Enzyme Inhib. Med. Chem. 2010, 25(6), 784-789

 

  • Erdaş, O.; Büyükbingol, E.; Alparslan, F.N.; Adejare, A. Modeling and Predicting Binding Affinity of Phencyclidine-Like Compounds Using Machine Learning Methods. J. Chemometrics 2010, 24, 1-13

 

  • Göker, H.; Coşkun, M.; Alp, Isolation and Identification of a New Acetildenafil Analogue Used To Adulterate A Dietary Supplement: Dimethylacetildenafil. Turk. J. Chem. 2010, 34, 157- 163

 

  • Hu, Q.; Negri, M.; Ölgen, S.; Hartmann, R.W. Role of Fluorine Substitution in Biphenyl Methylene Imidazole Type Cyp17 İnhibitors For The Treatment of Prostate Carcinoma. Med. Chem. 2010, 5 (6), 899-910

 

  • Karolak-Wojciechowska, J.; Szczesio, M.; Alper-Hayta, S.; Akı, E.; Yalçın, İ. Crystal Structure of 3,4-dihydro-3-oxo-6- ethoxycarbonyl-2H-1,4-benzoxazine-2-acetate, C15H17NO6, Kristallogr. NCS. 2010, 225, 531-532

 

  • Karolak-Wojciechowska, J.; Szczesio, M.; Ertan-Bolelli, T.; Akı, E.; Yalçın, İ. Crystal Structure of 4-fluoro-N-(2-hydroxy-4- nitrophenyl)benzamide, C13H9FN2O4, Z. Kristallogr. NCS. 2010, 225, 533-534

 

  • Kılıç, Z.; Şener, F.; İşgör, Y.G.; Çoban, T.; Ölgen, S. N-Substituted Indole-3-imine Derivatives and Their Amine Congeners: Antioxidant and Src Kinase Inhibitory Effects. Z. Naturforschung C 2010, 65c, 347-354

 

  • Kuş, C.; Sözüdönmez, F.; Can-Eke, B.; Çoban, T. Antioxidant and Antifungal Properties of Benzimidazole Derivatives. Zeitschrift für Naturforschung C 2010, 65C, 537-542

 

  • Ölgen, S.; Kaeßler, A.; Kılıç-Kurt, Z.; Jose, J.; Investigation of Aminomethyl Indole Derivatives as Hyaluronidase Inhibitors. Naturforschung C 2010, 65c, 445-450

 

  • Panicker, C.Y.; Varghese, H.T.; Ushakumari, l.; Ertan, T.;  Yıldız, İ.;  Granadeiro, C.M.; Nogueria, H.I.S.; Mary, Y.S. FT-IR, FT-Raman, SERS Spectra and Computational Calculations of 4-ethyl-N-(2’-hydroxy-5’-nitrophenyl)benzamide. Journal of Raman Spectroscopy 2010, 41, 381-390

 

  • Püsküllü, M.O.; Yıldız, S.; Göker, Synthesis and Antistaphylococcal Activity of N- substituted- 1Hbenzimidazole-sulphonamides, Archiv der Pharmazie 2010, 343,31- 39

 

  • Shirinzadeh, H.; Eren, B.; Gürer-Orhan, H.; Süzen, S.; Özden, S. Novel Indole-Based Analogs of Melatonin: Synthesis and İn Vitro Antioxidant Activity Studies. Molecules 2010, 15 (4), 2187-2202

 

  • Shirinzadeh, H.; Yilmaz, A.D.; Gümüştaş, M.; Süzen, S.; Özden, S.; Özkan, S.A. Electrochemical Behavior of Indole-3-carboxaldehyde izonicotinoyl hydrazones: Discussion on Possible Biological Behavior. Combinatorial Chemistry and High Throughput Screening 2010, 13 (7), 619-627

 

  • Süzen, S.; Özkan, S.A. Combination of Electrochemical, Spectrometric and other Analytical Techniques For High Throughput Screening of Pharmaceutically Active Compounds. Combinatorial Chemistry and High Throughput Screening 2010, 13 (7), 658-664

 

  • Yalçın, İ.; Akı, E.; Yıldız, İ.; Temiz-Arpacı, Ö. Antimicrobial Activity and Structure-Activity Relationships of Some Synthesized Benzazoles and Their Possible Med. Chem. Res. 2010, Suppl.:1, 19, S41

 

  • Yıldız, İ.; Bozdağ-Dündar, O. Three-Dimensional Common-Feature Hypotheses for Hypoglycemic Flavonyl-2,4thiazolidinedione Derivatives. Med. Chem. Res. 2010, 19, 211-219

 

  • Ateş-Alagöz, Z.; Sun, S.; Wallach J.; Adejare, A. Synthesis and Pharmacological Evaluations of Novel N-substitued bicyclo heptan-2-amines at NMDA Receptors. Chem. Biol. & Drug Design 2011, 78, 25-32

 

  • Bozdağ-Dündar, O.; Ertan, R.; Aboul-Enein, H.Y.; Kładna, A.; Kruk, I. Free Radical Scavenging Abilities of Flavonylthiazolidine-2,4-dione Compounds. Luminescence 2011, 26, 10-16

 

  • Bruno R.D.; Vasaitis, S.; Gediya, L.K.; Purushottamachar, P.; Godbole, A.M.; Ateş-Alagöz, Z.; Brodie, A.M.H.; Njar, V.C.O. Synthesis and Biological Evaluations of Putative Metabolically Stable Analogs of VN/124-1 (TOK-001) Analogs: Head to Head Anti-Tumor Efficacy Evaluation of VN/124-1(TOK-001) and Abiraterone in LAPC-4 Human Prostate Cancer Xenograft Model. Steroids 2011, 76, 1268-1279

 

  • Çetin, K.T.; Dinçer, S.; Ölgen, S. Synthesis of New Pyrrolo-[2,3-d]pyrimidine Derivatives as Src Kinase Inhibitors. Eur. J. Pharm. Sci. 2011, 44, suppl.1, 177-178

 

  • Daş-Evcimen, N.; Sarıkaya, M.; Gurkok, G.; Süzen, S. Evaluation of Rat Kidney Aldose Reductase İnhibitory Activity of Some N-Acetyl Dehydroalanine Derivatives. Medicinal Chemistry Research, 2011, 20 (4), 453-460

 

  • Gürkan, A.S.; Karabay, A.; Büyükbingol, Z.; Büyükbingol, E. Synthesis and Effects of Some Novel Tetrahydronaphthalene Derivatives on Proliferation and Nitric Oxide Production in Lipopolysaccharide Activated Raw 264.7 Macrophages. Eur. J. Med. Chem. 2011, 46, 468-479

 

  • Kaeßler, A.; Ölgen, S.; Jose, J. Autodisplay of Catalically Active Human Hyaluronidase hPH-20 and Testing of Enzyme Inhibitors. J. Pharm. Sci. 2011, 42(1-2), 138-147

 

 

  • Kılıç-Kurt, Z.; Ölgen, S. Synthesis of Novel Oxoindole Derivatives as Inhibitors of c-Src Tyrosine Kinase, Eur. J. Pharm. Sci. 2011, 44, suppl.1, 189

 

  • Ölgen, S.; İşgör, Y.G.; Kılıç-Kurt, Z.; Şener, F.; Çoban, T. Evaluation of Novel Aminomethylindole Derivatives as Src Kinase Inhibitors and Antioxidant Agents. Chemotheraphy 2011, 57, 1-6

 

  • Ölgen, S.; Kaessler, A.; Kılıç-Kurt, ; Jose, J. Structure-Activity Evaluation of N-benzyl-5-substituted indole-3-imine Derivatives and Their Amine Congeners as Bovine Testicular Hyaluronidase (BTH) Inhibitor. LDDD 2011, 8(8), 685-690

 

  • Ölgen, S. Design Src Kinase Inhibitors as a Therapeutic Approach for Cancer and Metastases, Eur. J. Pharm. Sci. 2011, 44, suppl.1, 18-19

 

  • Özden, ; Usta, F.; Altanlar, N.; Göker, H. Synthesis of Some New 1H- Benzimidazole- 2- carboxamido derivatives and their antimicrobial activitiy, J. Heterocyclic Chem. 2011, 48, 1317- 1322

 

  • Sheena Mary, Y.; Panicker, C.Y.;  Tresa Varghese, H.; Raju, K.; Ertan Bolelli, T.;  Yıldız, İ.; Granadeiro, M.C.;  Nogueira, H.I.S. Vibrational Spectroscopic Studies and Computational Study of 4-fluoro-N-(2’-hydroxy-4’nitrophenyl)phenylacetamide. Journal of Molecular Structure 2011, 994, 223-231

 

  • Shirinzadeh, H.; Altanlar, N.; Yucel, N., Özden, S.; Süzen, S. Antimicrobial Evaluation of İndole-Containing Hydrazone Derivatives. Zeitschrift fur Naturforschung – Section C Journal of Biosciences 2011, 66 C (7-8), 340-344.

 

  • Yüksel, N.; Baykara, M.; Shirinzadeh, H.; Süzen, S. Investigation of Triacetin Effect on İndomethacin Release From Poly(Methyl Methacrylate) Microspheres: Evaluation of Interactions Using FT-IR and NMR Spectroscopies. International Journal of Pharmaceutics 2011, 404 (1-2), 102-109

 

 

  • Ataei, S.; Yıldız, İ.; Karban, Ö.; Karabulut, M.; Dinç, E.; Tahiyeu, R.; Özbek, M.; ER, E.  Quantitative Analysis of Pantoprazole in Lyophilized Form by Using Hplc Method. J. Anal. Bioanal. Techniques 2012, 3(7), 102

 

  • Ataei, S.; Yıldız, İ.; Karban, Ö.; Karabulut, M.; Şimşek, H.; Dinç, E.; Tahiyeu, R.; Özbek, M.; ER, E.  High Performance Liquid Chromotographic Method For Determination of Clarithroycin in Lyophilized Form. J. Anal. Bioanal. Techniques 2012, 3(7), 103

 

  • Ateş-Alagöz, Z.; Coleman, N.; Martin, M.; Wan, A.; Adejare, A. In vitro Anticancer Properties of Novel Radiosensitizer Analogs. Chem. Biol. & Drug Design 2012, 80, 853-861

 

  • Ayhan-Kılcıgil, G.; Gürkan, S.; Çoban, T.; Özdamar, E.D.; Can-Eke, B. Synthesis and Evaluation of Antioxidant Properties of Novel 2-[2-(4-chlorophenyl) benzimidazole-1-yl]-N-(2-arylmethylene amino) acetamides and 2-[2-(4-chlorophenyl) benzimidazole-1-yl]-N-(4-oxo-2-aryl-thiazolidine-3-yl) acetamides-I. Chem. Bio. Drug Design 2012, 79, 869-877

 

  • Bolelli, K.; Yalçın, İ.; Ertan-Bolelli, T.; Özgen, S.; Kaynak-Onurdağ, F.; Yıldız, İ.; Akı, E.; Synthesis of novel 2-[4-(4- substituttedbenzamido/phenylacetamido)phenyl] benzothiazoles as antimicrobial agents. Chem. Res. 2012, 21, 3818-3825

 

  • Ezer, M.; Tatar-Yıldırım, L.; Bayro, O.; Verspohl, E.J.; Bozdağ-Dündar, O. Synthesis and Antidiabetic Activity of Morpholinothiazolyl-2,4-thiazolidindione Derivatives. J. Enzyme Inhib. Med. Chem. 2012, 27(3): 419-427

 

  • Göker,, Karaaslan, Ç.; Yıldız, S. Synthesis, Potent Antifungal and Antistaphylococcal Activities of Some New 2- Anilinobenzimidazoles, Z. Naturforsch. 2012, 67C, 486-494

 

  • Gürkan-Alp, A.S.; Mumcuoğlu, M.; Andaç, A.C.; Dayanç, E.; Atalay, R.; Büyükbingol, E. Synthesis, Anticancer Activities and Molecular Modeling Studies of Novel Indole Retinoid Derivatives. Eur. J. Med. Chem. 2012, 58, 346-354

 

  • Karataş, H.; Alp,; Yıldız, S.; Göker, H. Synthesis and Potent İn Vitro Activity of Novel 1H- Benzimidazoles as Anti- MRSA Agents. Chem Biol Drug Res. 2012, 80, 237-244

 

  • Karban, Ö.; Yıldız, İ.; Ataei, S.; Karabulut, M.; Dinç, E.; Tahiyeu, R.; Özbek, M.; ER, E.  High Performance Liquid Chromotographic Method For Determination of Azithromycin in Lyophilized Form. J. Anal. Bioanal. Techniques 2012, 3(7), 93

 

  • Kerimov, İ.; Ayhan-Kılcıgil, G.; Özdamar, E.D.; Can-Eke, B.; Çoban, T.; Özbey, S.; Kazak, C. Design, One-Pot and Microwave Assisted Synthesis of 2-Amino/5-aryl-1,3,4-oxadiazoles Bearing Benzimidazole Moiety as Antioxidant. Archiv der Pharmazie 2012, 345(7), 549-556

 

  • Sheena Mary, Y.; Raju, K.; Ertan Bolelli, T.;  Yıldız, İ.; Nogueira, H.I.S.; Granadeiro, C.M.; Alsenony, C.V.  FT-IR, FT-Raman, Surface Enhanced Raman Scattering and Computational Study of 2-(p-fluorobenzyl)-6-nitrobenzoxazole. Journal of Molecular Structure 2012, 1012, 22-30

 

  • Sheena Mary, Y.; Raju, K.; Yıldız, İ.; Temiz Arpacı, Ö.; Nogueira, H.I.S.; Granadeiro, C.M.; Alsenony, C.V. FT-IR, FT-Raman, SERS and Computational Study 3 of 5-ethylsulphonyl-2-(o-chlorobenzyl)benzoxazole.  Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 2012, 96, 617-625

 

  • Süzen, S.; Cihaner, S.S.; Çoban, T. Synthesis and Comparison of Antioxidant Properties of Indole-Based Melatonin Analogue Indole Amino Acid Derivatives. Chemical Biology and Drug Design 2012, 79 (1), 76-83

 

  • Taşkın,T.; Yılmaz, S.; Yıldız, İ.; Yalçın, İ.; Akı, E. Insight into Eukaryotic Topoisomerase II-Inhibiting Fused Heterocyclic Compounds in Human Cancer Cell Lines by Molecular Docking. SAR and QSAR in Environmental R 2012, 23(3–4), 345–355

 

  • Tunçbilek, M.; Bilget Güven, E.; Önder, T.; Çetin Atalay, R. Synthesis of Novel 6-(4-Substituted piperazine-1-yl)-9-(β-Dribofuranosyl)purine Derivatives, Which Lead to Senescence-Induced Cell Death in Liver Cancer Cells. J. Med. Chem.  2012, 55(7), 3058-3065

 

  • Yılmaz, A.D.; Çoban, T.; Süzen, S. Synthesis and Antioxidant Activity Evaluations of Melatonin-Based Analogue Indole Hydrazide/ Hydrazone Derivatives. J. Enzyme Inhib. Med. Chem. 2012, 27 (3), 428-436

 

  • Alp, ; Coşkun, M.; Göker, H.  Isolation and identification of a new Sildenafil analogue adulterated in Energy Drink : Propoxyphenyl Sildenafil J. Pharm. & Biomed. Anal. 2013, 72, 155- 158

 

  • Altıntop, M.D.; Gürkan-Alp, A.S.; Özkay, Y.; Kaplancıklı, Z.A. Synthesis and Biological Evaluation of A Series of Dithiocarbamates as New Cholinesterase Inhibitors. Pharm. Chem. Life Sci. 2013, 346 (8), 571-576

 

 

  • Ateş-Alagöz, Z.; Adejare, A. NMDA Receptor Antagonists for the Treatment of Depression, Pharmaceuticals, Special Issue, NMDA Receptor Antagonists for the Treatment of CNS Disorders 2013, 6 (4), 480-499

 

  • Ateş-Alagöz, Z.; Antioxidant Activities of Retinoidal Benzimidazole or Indole Derivatives in In Vitro Model Systems, Current Medicinal Chemistry,  Special Issue, Chemistry and Biology of Antioxidants 2013, 20 (36), 4633-4639

 

 

 

  • Bhagyasree, J.B.; Varghese, H.T.; Panicker, C.Y.; Samuel, J.; Van Alsenoy, C.; Yılmaz, S.; Yıldız, İ.; Akı, E. Quantum Mechanical and Spectroscopic (FT-IR, FT-Raman, 1H NMR and UV) Investigations of 2-(p-nitrobenzyl)benzoxazole. Journal of Molecular Structure 2013, 1046, 92-100

 

  • Bhagyasree, J.B.; Varghese, H.T.; Panicker, C.Y.; Samuel, J.; Van Alsenoy, C.; Bolelli, K.; Yıldız, İ.; Akı, E. Vibrational Spectroscopic (FT-IR, FT-Raman, 1H NMR and UV) Investigations and Computational Study of 5-nitro-2-(4-nitrobenzyl) benzoxazole. Spectrochimica Acta – Part A: Molecular and Biomolecular Spectroscopy 2013, 102, 99-113

 

  • Bhagyasree, J.B.; Samuel, J.; Varghese, H.T.; Panicker, C.Y.; Arısoy, M.; Temiz-Arpacı, Ö. Synthesis, FT-IR Investigation and Computational Study of 5-[(4-Bromophenyl)acetamido]-2-(4-tert-butylphenyl) benzoxazole. Spectrochimica Acta – Part A: Molecular and Biomolecular Spectroscopy, 2013, 115, 79-91

 

  • Borges, F.; Saso, L.; Garrido, J.; Süzen, S. Synthesis, Evaluation and Pharmacological Applications of Antioxidants-Part 2. Current Medicinal Chemistry 2013, 20 (37), 4647

 

  • Borges, F.; Saso, L.; Garrido, J.; Süzen, S. Synthesis, Evaluation and Pharmacological Applications of Antioxidants-Part 1. Current Medicinal Chemistry 2013, 20 (36), 4435

 

  • Can, A.; Yıldız, İ.; Güvendik, G. The Determination of Toxicities of Sulphonylurea and Phenylurea Herbicides with Quantitative Structure–Toxicity Relationship (QSTR) Studies.  Environmental Toxicology and Pharmacology 2013, 35, 369-379

 

  • Ceylan-Ünlüsoy, M.; Kazak, C.; Bayro, O.; Verspohl, E.J.; Ertan, R.; Bozdağ-Dündar, O. Synthesis and Antidiabetic Activity of 2,4-Thiazolidindione, Imidazolidinedione and  2-Thioxo-Imidazolidine-4-one Derivatives Bearing 6-Methyl Chromonyl Pharmacophore. Enzyme Inhib. Med. Chem. 2013, 28(6): 1205-1210

 

  • Coleman, N.; Ateş-Alagöz, Z.; Gaye, B.; Farbaniec, M.; Sun, S.; Adejare, A. Toxicity Studies on Novel N-substituted bicyclo-heptan-2-amines at NMDA Receptors. Pharmaceuticals, Special Issue, NMDA Receptor Antagonists for the Treatment of CNS Disorders 2013, 6(4), 536-545

 

  • Daş-Evcimen, N.; Sarıkaya, M.; Gürkan, S.; Bozdağ-Dündar, O. Aldose Reductase Inhibitory Potential of Several Thiazolyl-thiazolidine-2,4-diones. Letters in Drug Design and Discovery 2013, 10(5), 415-419

 

  • Dinçer, S.; Cetin, K.T.; Onay-Beşikci, A.; Ölgen, S. Synthesis, Biological Evaluation and Docking Studies of New Pyrrolo-[2,3-d] Pyrimidine Derivatives as Src Family-Selective Tyrosine Kinase Inhibitors. J. Enzym. Inhib. Med. Chem. 2013, 28(5), 1080-1087

 

  • Erdas, O.; Andac A.C.; Gürkan-Alp, A.S.; Alparslan, F.N.; Büyükbingol, E. Compressed Images for Affinity Prediction (CIFAP): A Study on Predicting Binding Affinities for Checkpoint Kinase 1 Protein Inhibitors. J. Chemometrics 2013, 27,  155-164

 

  • Kaplan-Özen, Ç.; Tekiner-Gülbaş, B.; Foto, E.; Yıldız, İ.; Diril, N.; Akı, E.; Yalçın, İ. Benzothiazole Derivatives as Human DNA Topoizomerase IIα Med. Chem. Res. 2013, 22(12), 5798-5808

 

  • Karaaslan, Ç.; Kadri, H.; Çoban, T.; Süzen, S.; Westwell, A.D. Synthesis and Antioxidant Properties of Substituted 2-Phenyl-1H-Indoles. Bioorg. Med. Chem. Lett. 2013, 23, 2671-2674

 

  • Kılıç-Kurt, Z.; Aydın, D.; İşgör, Y.G.; İşgör, B.S.; Ölgen, S. Synthesis and Biological Study of Novel Indole-3-imine-2-on Derivatives as Src Kinases and Glutathione S-Transferase Inhibitor. LDDD 2013, 10 (1), 19-26

 

  • Kılıç-Kurt, Z.; Onay-Beşikci, A.; Ölgen, S. Synthesis, Biological and Computational Evaluation of Novel Oxindole Derivatives as Inhibitors of Src Family Kinases, LDDD 2013, 10 (8), 713-718

 

  • Ölgen, S.; Gratz, A.; Kılıç Kurt, Z.; Jose, J.  Molecular Modeling Based Approach and In Vitro Assay of N-Substituted Indole-2 and 3-Carboxamide Derivatives as Human Protein Kinase CK2 Inhibitor. Acta Chimica Slovenica 2013, 60, 628-635

 

  • Ölgen, S.; Bakar, F.; Aydın, S.; Nebioğlu, D.; Nebioğlu, S. Synthesis of New İndole-2- Carboxamide and 3-Acetamide Derivatives and Evaluation Their Antioxidant Properties. J. Enzym. Inhib. Med. Chem. 2013, 28 (1), 58-64

 

  • Purushottamachar, P.; Godbole, A.M.; Gediya, L.; Martin, M.; Vasaitis, T.; Kwegyir-Afful, A.; Ateş-Alagöz, Z.; Njar, V.C.O. Systematic Structure Modifications of Multi-target Prostate Cancer Clinical Candidate Galeterone to Produce Novel Androgen Receptor Down-regulating Agents as an Approach to Treatment of Advanced Prostate Cancer. Journal of Medicinal Chemistry, 2013, 56 (12), 4880-4898

 

  • Püsküllü, M.O.; Tekiner, B.; Süzen, S. Recent Studies of Antioxidant Quinoline Derivatives. Mini-Reviews in Medicinal Chemistry 2013, 13 (3), 365-372

 

  • Süzen, S.; Tekiner-Gülbaş, B.; Shirinzadeh, H.; Uslu, D.; Gürer-Orhan, H.; Gümüştaş, M., Özkan, S.A. Antioxidant Activity of Indole-Based Melatonin Analogues In Erythrocytes and Their Voltammetric Characterization. Enzyme Inhib. Med. Chem. 2013, 28 (6), 1143-1155

 

  • Süzen, S.; Saso, L. Antioxidant Heterocyclic Compounds in Drug Discovery and Medicinal Chemistry. Mini-Reviews in Medicinal Chemistry 2013, 13 (3), 317

 

  • Süzen, S., Melatonin and Synthetic Analogs as Antioxidants. Current Drug Delivery 2013, 10 (1), 71-75

 

  • Tekiner-Gülbaş, B.; Westwell, A.D.; Süzen, S. Oxidative Stress in Carcinogenesis: New Synthetic Compounds with Dual Effects Upon Free Radicals and Cancer. Current Medicinal Chemistry 2013, 20 (36), 4451-4459

 

 

  • Wannberg, J.; Wallinder, C.; Ünlüsoy, M.; Sköld, C.; Larhed, M. One-Pot, Two-Step, Microwave-Assisted Palladium-Catalyzed Conversion of Aryl Alcohols to Aryl Fluorides Via Aryl Nonaflates. Journal of Organic Chemistry 2013, 78, 4184-4189

 

  • Yılmaz, S.; Yalçın, İ.; Kaynak-Onurdağ, F.; Özgen, S.; Yıldız, İ.; Akı, E. Synthesis and In vitro Antimicrobial Activity of Novel 2-(4- (Substituted-carboxamido)benzyl/ phenyl)benzothiazoles, Croatica Chemical Acta 2013, 86(2), 223-231

 

  • Alp, M.; Göker, A.H.; Altanlar N. Synthesis and antimicrobial activity of novel 2-[4-(1H-benzimidazol-1-yl)phenyl]-1H-benzimidazoles.  J. Chem. 2014, 38, 152-156

 

  • Alp, M.; Göker, H.; Ozkan, T.; Sunguroğlu, A.  Synthesis and cytotoxic evaluation of novel N-substituted amidino-1-hydroxybenzimidazole derivatives.  Archives of Pharmacal Research 2014, 37(5), 580-587

 

  • Akı-Yalçın, E.; Ertan-Bolelli, T.; Taşkın-Tok, T.; Öztürk, Ö.; Ataei, S.; Özen, C.; Yıldız, İ.; Yalçın, İ. Evaluation of Inhibitory Effects of Benzothiazole and 3-Amino-benzothiazolium Derivatives on DNA Topoisomerase II by Molecular Modeling Stu SAR and QSAR in Environmental Research 2014, 25(8), 637-649

 

 

  • Ayhan-Kilcigil, G.; Kuş, C.; Çoban,T.; Özdamar, E.D.; Can-Eke, B. Identification of a Novel Series of N-Phenyl-5-[(2-phenylbenz-imidazol-1-yl)methyl]-1,3,4-oxadiazol-2-amines as Potent Antioxidants and Radical Scavengers.  Pharm. Chem. Life Sci. 2014, 347, 276-282

 

  • Berczynski, P.; Duchnik, E.; Kruk, I.; Piechowska, T.; Aboul-Enein, H.Y.; Bozdağ-Dündar, O.;  Ceylan-Ünlüsoy, M. 6-Methyl 3-chromonyl 2,4-thiazolidinedione/2,4-imidazolidinedione/2-thioxoimidazolidine-4-one Compounds: Novel Scavengers of Reactive Oxygen Species.  Luminescence 2014, 29(4), 367-373

 

  • Berczynski, P.; Kładna, A.; Piechowska, T.; Kruk, I.; Bozdağ-Dündar, O.; Aboul-Enein, H.Y.;  Ceylan-Ünlüsoy, M.; Ertan, R. Studies on The Antioxidant Activity of Some Thiazolidinedione, Imidazolidinedione and Rhodanine Derivatives Having a Flavone Core. Luminescence 2014, 29(8), 1107-1112

 

  • Ertan-Bolelli, T.; Musdal, Y.; Bolelli, K.; Yılmaz, S.; Aksoy, Y.; Yıldız, İ.; Akı-Yalçın, E.; Yalçın, İ. Synthesis, Biological Evaluation of 2-Substituted-5-(4-nitrophenylsulfonamido) benzoxazoles as Human GST P1-1  Inhibitors and Description of the Binding Site Features. ChemMedChem 2014, 9(5), 984-992

 

  • Kładna, A.; Berczynski, P.; Piechowska, T.; Kruk, I.; Aboul-Enein, H.Y.; Ceylan-Ünlüsoy, M.; Verspohl, E.J.; Ertan, R. Studies on The Antioxidant Activities of Some New Chromone Compounds. Luminescence 2014, 29(7), 846-853

 

  • Yılmaz, A.D.; Karaaslan Ç., Shirinzadeh, H.; Süzen S.; Özcan S.; Gürer-Orhan, H. New Antioxidant Drug Development Studies on Neurohormone Melatonin and Synthetic Analogues. Academic Journal of Science 2014, 03(02), 51-56

 

  • lmaz, S.; Altınkanat-Gelmez, G.; Bolelli, K.; Guneser-Merdan, D.; Over-Hasdemir, M.U.; Yıldız, I.; Akı-Yalçın, E.; Yalçın, İ. Pharmacophore Generation of 2- Substituted Benzothiazoles as AdeABC Efflux Pump Inhibitors in A. Baumannii. SAR and QSAR in Environmental Research 2014, 25(7), 551-563

 

  • Zilifdar, F.; Alper-Hayta, S.; Yılmaz, S.; Kaplan-Özen, Ç.; Foto, E.; Aydoğan, Z.; Yıldız, İ.; Akı, E.; Yalçın, İ.; Diril, N. Genotoxic Potentials and Eukaryotic DNA Topoisomerase I Inhibitory Effects of Some Benzoxazine Derivatives. Med. Chem. Res. 2014, 23(1), 480-486

 

  • Alp, M.; Gürkan-Alp, A.S.; Özkan, T.; Sunguroğlu, A. Synthesis and Anticancer Evaluation of Novel 5-(4-Methylpiperazin-1-yl)-2-Phenyl-1H-Benzimidazole Derivatives. Zeitschrift für Naturforschung C – A Journal of Biosciences [Online early access]. DOI:1515/znc-2014-4189. 2015

 

  • Alp, A.S.; Kılcıgil, G.; Özdamar, E.D.; Çoban, T.; Eke, B. Synthesis and Evaluation of Antioxidant Activities of Novel 1,3,4-oxadiazole and Imine Containing 1H-benzimidazoles. Turkish Journal of Chemistry 2015, 39, 42-53

 

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